Exploiting C–H borylation for the multidirectional elaboration of 2-halopyridines
Regioselectively polysubstituted pyridines can be efficiently accessed from 2-halopyridines via a sequence involving C–H borylation, Suzuki-Miyaura cross-coupling and nucleophilic aromatic substitution chemistry.
Reuven, Jonathan A.,Salih, Omar A.,Sadler, Scott A.,Thomas, Carys L.,Steel, Patrick G.
The present invention relates to compounds of the formula wherein R1 to R8 are as defined in the description and claims, and pharmaceutically acceptable salts thereof. The compounds are useful for the treatment and/or prophylaxis of
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(2008/06/13)
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