Nucleophilic ring opening of aziridines with amines under catalyst- and solvent-free conditions
The aza-addition of aziridines to obtain vicinal-diamines was achieved under catalyst- and solvent-free conditions for the first time. Various aryl, alkyl and meso-bicyclic aziridines with a Ts-protecting group were tolerated, and aromatic amine-nucleophi
Reactions with Aziridines, 38. On the Regioselectivity of the Nucleophilic Ring Opening of Activated 2-Phenylaziridines
The ring of 1-mesyl (1c) and 1-(phenylcarbamoyl)-2-phenylaziridine (1d) is opened between N and C-2 (benzylic effect) by some nucleophiles in high yields.
Onistschenko, Andreas,Buchholz, Berthold,Stamm, Helmut
p. 2678 - 2680
(2007/10/02)
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