1,2-disubstituted indole, azaindole and benzimidazole derivatives possessing amine moiety: A novel series of thrombin inhibitors
A novel series of 1,2-disubstituted indole, azaindole and benzimidazole derivatives possessing an amine moiety was identified as thrombin inhibitors. An indole with basic diamine moieties (12a) was the most potent thrombin inhibitor in the series with K(ass) = 197 x 106 L/mol. (C) 2000 Elsevier Science Ltd.
Takeuchi, Kumiko,Bastian, Jolie A.,Gifford-Moore, Donetta S.,Harper, Richard W.,Miller, Shawn C.,Mullaney, Jeffrey T.,Sall, Daniel J.,Smith, Gerald F.,Zhang, Minsheng,Fisher, Matthew J.
p. 2347 - 2351
(2007/10/03)
Preparation of new fluorine containing 2-phenylindole derivatives as antifertility agents
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Joshi,Jain,Garg
p. 388 - 390
(2007/10/02)
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