- Based on isoxazole substitution of benzamide derivatives and anti-prostate cancer drug applications
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The present invention discloses a class (I), formula (II) structure based on isoxazole substituted benzamide derivatives and antiprostate cancer drug applications, such isoxazole substituted benzamide derivatives, can effectively inhibit the activity of a
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Paragraph 0065; 0073-0074
(2022/01/10)
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- Piperazine derivatives and the use thereof as medicament
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The present inventions relate to substituted piperazine derivatives of general formula (I) and to the manufacture of said compounds, pharmaceutical compositions comprising a compound according to general formula (I), and the use of said compounds for the treatment of various medical conditions related to glycine transporter-1 (GlyT1).
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Paragraph 0223; 0224; 0225; 0226
(2015/04/21)
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- PIPERAZINE DERIVATIVES AND THE USE THEREOF AS MEDICAMENT
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The present inventions relate to substituted piperazine derivatives of general formula (I) and to the manufacture of said compounds, pharmaceutical compositions comprising a compound according to general formula (I), and the use of said compounds for the treatment of various medical conditions related to glycine transporter-1 (GlyT1).
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Page/Page column 50; 51
(2015/05/05)
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- Photoactive azole pesticides
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Oxazole and thiazole compounds of the following formula are photodynamic insecticides and acaricides as well as nematicides: STR1 wherein W is selected from O and S; R2 is selected from optionally substituted thienyl and optionally substituted phenyl; R4 is selected from hydrogen, lower alkyl, lower haloalkyl, thienyl, tri(lower alkyl)silyl, and optionally substituted phenyl; R5 is selected from optionally substituted thienyl and optionally substituted phenyl; at least one of R2 and R5 is an optionally substituted thienyl group, and R4 is other than hydrogen when R4 and R5 are each unsubstituted phenyl or thienyl.
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