Synthesis and evaluation of a 11C-labelled angiotensin II AT2 receptor ligand
Three 11C-radiolabelled high-affinity nonpeptide AT2 receptor-selective ligands were synthesized and one of these was evaluated as positron emission tomography (PET) tracer. The labelling reaction was performed via palladium(0)-media
Selective angiotensin II AT2 receptor agonists: Benzamide structure-activity relationships
In the investigation of the structure-activity relationship of nonpeptide AT2 receptor agonists, a series of substituted benzamide analogues of the selective nonpeptide AT2 receptor agonist M024 have been synthesised. In a second ser