One-pot synthesis of ureido peptides and urea-tethered glycosylated amino acids employing deoxo-fluor and TMSN3
A facile one-pot procedure for the synthesis of urea-linked peptidomimetics and neoglycopeptides under Curtius rearrangement conditions employing Deoxo-Fluor and TMSN3 is described. The method is efficient and circumvents the isolation of acyl