Towards to hENT1-nucleoside transporter selective imaging agents. Synthesis and in vitro evaluation of the radiolabeled SAENTA analogues
Three new potential hENT1 inhibitors suitable for labeling with PET/SPECT radioisotopes were prepared from an advanced intermediate 4. They were tested for their capability to inhibit binding of SAENTA-fluorescein to HL60 leukemia cells in flow
Zlatopolskiy, Boris D.,Morgenroth, Agnieszka,Urusova, Elizaveta A.,Dinger, Cornelia,Kull, Thomas,Pape, Manuela,Glatting, Gerhard,Reske, Sven N.