DIASTEREOSELECTIVE CHLOROCYCLOFUNCTIONALIZATION OF N-ALLYLIC TRICHLOROACETAMIDES: SYNTHESIS OF AN ANALOGUE AND POTENTIAL PRECURSOR OF RP49532
Treatment of (E)-N-cinnamyl trichloroacetamide with hypochlorous acid yielded trans-dihydro-oxazine 8 which was easily hydrolyzed to (+/-)-erythro-β-chloro-γ-hydroxy-γ-phenyl-propanamine 2.Applied to the imidazole series, this chlorocyclization gave 15, a
Commercon, A.,Ponsinet, G.
p. 3871 - 3874
(2007/10/02)
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