Small-Molecule Choline Kinase Inhibitors as Anti-Cancer Therapeutics
Small molecule choline kinase inhibitors having the following formula: are provided herein. Also provided herein are pharmaceutical compositions containing Formula I compounds, together with methods of treating cancer, methods of inhibiting choline kinase enzymatic activity, and methods of treating tumors by administering an effective amount of a Formula I compound.
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Page/Page column 19; 27-28
(2011/10/31)
New derivatives of 1,2,4-triazole
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Russo,Ghelardoni
p. 128 - 139
(2007/10/08)
On various derivatives of 2-(o.ethoxyphenyl)-1,3,4-oxadiazole 5-mercapto-subtituted