5-Halobenzothiophene analogues of melatonin: Synthesis and affinity for mt1 and MT2 receptors in man
A novel series of melatonin analogues based on the benzothiophene nucleus is described. In these compounds the methoxy group was replaced by electron-attracting groups such halogens (Br and Cl) with the aim of supplementing structure-affinity relationship
This invention provides novel 5-HT1Fagonists of formula where X, Y, Z,and R are defined in the specification, which are useful for the prevention and treatment of migraine and associated disorders.
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(2008/06/13)
Pharmacologically active benzo[b]thiophen derivatives. 8. Benzo[b]thiophen analogues of tryptophan and alpha-methyltryptophan, and some of their 5-substituted derivatives.
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Chapman,Scrowston,Westwood
p. 1855 - 1858
(2007/10/08)
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