- TETRAHYDROPYRROLOTHIAZINE COMPOUNDS
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The present invention provides compounds of Formula I: wherein A is selected from the group consisting of; R1 is H or F; R2 is H, —CH2OH, C1-C3 alkyl, R3 is H, F, or CN; R4 is H, F; or CN; and R5 is H, —CH3, or —OCH3; or a pharmaceutically acceptable salt thereof.
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Paragraph 0089; 0090
(2013/10/08)
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- Cross-metathesis of N-alkenyl peptoids with O- or C-allyl glycosides
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Cross-metathesis of several N-alkenyl-containing oligoglycines derivatives (peptoids) with protected O or C-allyl glycosides of N- acetylglucosamine, galactose, and mannose using Grubbs' ruthenium benzylidene catalyst (Cy3P)2Cl2Ru=CHPh (1) has been achieved in 40 to 52% yields.
- Hu, Yun-Jin,Roy, Rene
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p. 3305 - 3308
(2007/10/03)
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- Synthesis and reactions of 9,10-diazatetracyclo-[6.3.0.0.4,110.5.9]undecanes
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The tandem 1,3-dipolar cycloaddition between sydnones and 1,5-cyclooctadiene provides 9,10-diazatetracyclo[6.3.0.0.4,110.5,9]undecanes (the Weintraub reaction) in modest to good yields.
- Gribble, Gordon W.,Hirth, Bradford H.
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p. 719 - 726
(2007/10/03)
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