2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]-naphthalenyl derivatives with antipsychotic activity
Compounds of the Formula (I): are useful in the treatment of disorders associated with brain dopamine dysregulation.
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(2008/06/13)
2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]-naphthalenyl derivatives with antipsychotic activity
Compounds of the Formula (I): are useful in the treatment of disorders associated with dopamine dysregulation.
-
(2008/06/13)
New generation dopaminergic agents. Part 8: Heterocyclic bioisosteres that exploit the 7-OH-2-(aminomethyl)chroman D2 template
Based on the 7-OH-2-(aminomethyl)chroman dopamine D2 template (2) is described the preparation and resolution of two bioisosteric analogues. The benzimidazol-2-one derivative (6) had similar affinity to the known indolone derivative (4).
Mewshaw, Richard E.,Zhao, Rulin,Shi, Xiaojie,Marquis, Karen,Brennan, Julie A.,Mazandarani, Hossein,Coupet, Joseph,Andree, Terrance H.
p. 271 - 274
(2007/10/03)
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