- 1 -HYDROXY-BENZOOXABOROLES AS ANTIPARASITIC AGENTS
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Provided are compounds useful for controlling endoparasites both in animals and agriculture. Further provided are methods for controlling endoparasite infestations of an animal by administering an effective amount of a compound as described above, or a pharmaceutically acceptable salt thereof, to an animal, as well as formulations for controlling endoparasite infestations using the compounds described above or an acceptable salt thereof, and an acceptable carrier. The claimed compounds are described by the following Markush formula:A typical example for a compound according to above formula is: A typical example for a compound according to above formula is:
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Page/Page column 57
(2014/10/03)
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- Preparative synthesis of vanillin and vanillal alkanoates
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Procedures for preparing vanillin and vanillal alkanoates were developed.
- Dikusar,Vyglazov,Moiseichuk,Zhukovskaya,Kozlov
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p. 120 - 124
(2007/10/03)
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- Vanillal esters in reaction with 2-naphthylamine and 1,3-diketones
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Analogs of natural alkaloids of acridone series, derivatives of 4-(9-alkyl-11-oxo-7,8,9,10,1,12-hexahydro-benzo[a]acridin-12-yl) and 4-(12-oxo-12H-benzo[f]indeno[1,2-b]quinolin-13-yl)2-ethoxyphenyl carboxylates were synthesized by a three-component conden
- Kozlov,Basalaeva,Dikusar
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p. 1637 - 1646
(2007/10/03)
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- Reactions of vanillin and vanillal esters with 6-quinolylamine and phenidone
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Previously unknown 2-methoxy(or ethoxy)-4-(11-oxo-9-phenyl-7,8,9,10,11,12- hexahydrobenzo[b][4,7]phenanthrolin-12-yl)phenyl esters of carboxylic acids were prepared by ternary condensation of vanillin or vanillal alkanoates with 6-quinolylamine and Phenid
- Gusak,Kozlov
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p. 1562 - 1565
(2007/10/03)
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- Synthesis and evaluation of novel thiazolidine derivatives as thromboxane A2 receptor antagonists
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A series of 3-benzoyl or 3-phenylsulfonyl-2-substituted thiazolidine derivatives were synthesized, and evaluated for their thromboxane A2 (TXA2) receptor-antagonizing effect on (15S)-15-hydroxy-11α,9α- (epoxymethano)prosta-5(Z),13(E)-dienoic acid (U-46619)-induced aggregation of rabbit platelet-rich plasma (PRP). A simple 2-arylthiazolidine derivative, 3- benzoyl-2-(4-hydroxy-3-methoxyphenyl)thiazolidine (5a), showed mild TXA2 receptor antagonist activity. Modification of 5a led to 2-chloro-4-[3-(4- chlorophenylsulfonyl)thiazolidin-2-ylmethyl]phenoxyaretic acid (29d), which showed 10 times more potent TXA2 receptor antagonist activity than 5a.
- Sato,Kawashima,Goto,Yamane,Chiba,Jinno,Satake,Imanishi,Iwata
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p. 521 - 529
(2007/10/02)
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