Journal of Medicinal Chemistry p. 1663 - 1668 (1986)
Update date:2022-07-31
Topics:
Wouters, Walter
Janssen, Cornelus G. M.
Dun, Jacky Van
Thijssen, Jos B. A.
Laduron, Pierre M.
<3H>-7-Aminoketanserin (7-amino-3-<2-<4-(2-tritio-4-fluorobenzoyl)-1-piperidinyl>ethyl>-2,4-(1H,3H)-quinazolinedione), an amino derivative of the selective serotonin-S2 antagonist ketanserin, was synthesized and tested for in vitro labeling of serotonin-S
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(1985)