Bioorganic and Medicinal Chemistry Letters p. 3156 - 3161 (2006)
Update date:2022-08-02
Topics:
Penning, Thomas D.
Khilevich, Albert
Chen, Barbara B.
Russell, Mark A.
Boys, Mark L.
Wang, Yaping
Duffin, Tiffany
Engleman, V. Wayne
Finn, Mary Beth
Freeman, Sandra K.
Hanneke, Melanie L.
Keene, Jeffery L.
Klover, Jon A.
Nickols, G. Allen
Nickols, Maureen A.
Rader, Randall K.
Settle, Steven L.
Shannon, Kristen E.
Steininger, Christina N.
Westlin, Marisa M.
Westlin, William F.
We describe a series of pyrazole and isoxazole analogs as antagonists of the αvβ3 receptor. Compounds showed low to sub-nanomolar potency against αvβ3, as well as good selectivity against αIIbβ3<
View Morewebsite:http://www.jairadhesales.com
Contact:0091-79-26431096
Address:309 Harikrupa Tower,Nr old Sharda Mandir Char Rasta,Ellisbridge
Contact:+86-20-32051076
Address:1105,Building A, International Business Incubator,Science City
Shanghai Yudiao Chemistry Technology Co.,Ltd
Contact:0086-18964703211
Address:Building NO.5, NO.218,Rongtian Road,ganxiang town,Jinshan District,shanghai,201518,china
SHENZHEN PENGCHENG REDSTAR INDUSTRY CO.,LTD
Contact:+86-755-82412922
Address:Room 8066, East Block, Square City, Jiabin Road, Luohu District
Guangxi Nanning Guangtai Agriculture Chemical Co.,Ltd
Contact:+86-771-2311266
Address:Room703,Building12, Software Park Phase II,NO.68,Keyuan Road,Nanning City,Guangxi,China
Doi:10.1039/j39710003415
(1971)Doi:10.1016/S0022-328X(00)99521-4
(1986)Doi:10.1002/jps.2600600816
(1971)Doi:10.1002/1521-3773(20010302)40:5<952::AID-ANIE952>3.0.CO;2-S
(2001)Doi:10.1016/j.tetasy.2003.09.023
(2003)Doi:10.1016/S0960-894X(03)00474-8
(2003)