Journal of labelled compounds and radiopharmaceuticals p. 757 - 772 (1997)
Update date:2022-08-04
Topics:
Emond
Boazi
Duchene
Chalon
Besnard
Guilloteau
Frangin
The synthesis of (E)-N-(3-iodoprop-2-enyl)-2β-carbomethoxy-3β-(3',4'-dichlorophenyl) nortropane (β-CDIT) and its radioiodinated analogues is described. Three different synthetic methods are reported for the preparation of (E)-N-[3-(tributylstannyl)-2-enyl]-2β-carbomethoxy-3β-(3', 4'-dichlorophenyl) nortropane, which was iododestannylated for the preparation of the corresponding iodinated derivative. We also report the radiolabelling of β-CDIT with 125I or 123I that could be used for in vitro and in vivo exploration of the dopamine transporter.
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