139548-35-9Relevant articles and documents
The synthesis of several tritiated non-nucleoside, HIV-1 reverse transcriptase inhibitors
Hamill, Terence G.,Brenner, Nancy J.,Eng, Wai-Si,Burns, H. Donald
, p. 319 - 327 (2007/10/03)
The synthesis of three tritiated reverse transcriptase inhibitors is described herein. These compounds contained the benzoxazole ring linked to a 2-pyridinone ring by an aminomethylene group. The tritiated compounds were synthesized by hydrogenolysis of bromobenzoxazole precursors. The final tritiated compounds had specific activities ranging from 3-10 Cl/mmol.