173974-87-3Relevant articles and documents
Direct and Regioselective C(sp 3)-H Bond Fluorination of 2-Alkylazaarenes with Selectfluor
Le Guen, Clothilde,Mazzah, Ahmed,Penhoat, Ma?l,Melnyk, Patricia,Rolando, Christian,Chausset-Boissarie, La?titia
, p. 1157 - 1162 (2021)
Herein, a regioselective and direct monofluorination strategy of pyridylic and quinolinic C(sp 3)-H bonds was developed under transition-metal-free conditions with Selectfluor. The reaction was performed under smooth conditions and afforded fluorinated azahetero cycles including 2-methylpyridines and -quinolines in moderate to good yields.
PROCESSES FOR FLUORINATION
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Paragraph 0188, (2020/03/05)
The present technology relates to fluorination reactions. Specifically, processes useful for making the fungicide compound, DFT are disclosed. More broadly, also disclosed herein are processes useful for deoxyfluorination at the α-aromatic position of a given compound.
Reaction of N-fluoropyridinium fluoride with isonitriles and diazo compounds: A one-pot synthesis of (pyridin-2-yl)-1H-1,2,3-triazoles
Kiselyov, Alexander S.
, p. 2631 - 2634 (2007/10/03)
Reaction of N-fluoropyridinium fluoride generated in situ with a series of isonitriles and diazo compounds led to the formation of the corresponding (pyridine-2-yl)-1H-1,2,3-triazoles in good yields (37-59%). Best outcome was consistently achieved with bo
