191793-72-3Relevant articles and documents
Fluorinated peptides incorporating a 4-fluoroproline residue as potential inhibitors of HIV protease
Tran, Thanh Thu,Patino, Nadia,Condom, Roger,Frogier, Tea,Guedj, Roger
, p. 125 - 130 (2007/10/03)
N-Fmoc-4-fluoro-L-proline methyl ester was prepared as an attractive synthon for both solid and solution phase peptide synthesis. Its use for the synthesis of Fmoc-Phe-Pro(F)-OMe and Fmoc-Pro(F)-Val-Val-OMe is presented. Direct fluorination with DAST of a