103906-30-5Relevant articles and documents
Synthesis of long-chain amide analogs of the cannabinoid CB1 receptor antagonist N-(piperidinyl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl- 1H-pyrazole-3-carboxamide (SR141716) with unique binding selectivities and pharmacological activities
Thomas, Brian F.,Francisco, Ma. Elena Y.,Seltzman, Herbert H.,Thomas, James B.,Fix, Scott E.,Schulz, Anne-Kathrin,Gilliam, Anne F.,Pertwee, Roger G.,Stevenson, Leslie A.
, p. 5463 - 5474 (2005)
An extended series of alkyl carboxamide analogs of N-(piperidinyl)-5-(4- chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl- 1H-pyrazole-3-carboxamide (SR141716; 5) was synthesized. Each compound was tested for its ability to displace the prototypical cannabin
