1225208-12-7Relevant articles and documents
The identification of a selective dopamine D2 partial agonist, D3 antagonist displaying high levels of brain exposure
Holmes, Ian P.,Blunt, Richard J.,Lorthioir, Olivier E.,Blowers, Stephen M.,Gribble, Andy,Payne, Andrew H.,Stansfield, Ian G.,Wood, Martyn,Woollard, Patrick M.,Reavill, Charlie,Howes, Claire M.,Micheli, Fabrizio,Fabio, Romano Di,Donati, Daniele,Terreni, Silvia,Hamprecht, Dieter,Arista, Luca,Worby, Angela,Watson, Steve P.
body text, p. 2013 - 2016 (2010/09/18)
The identification of a highly selective D2 partial agonist, D3 antagonist tool molecule which demonstrates high levels of brain exposure and selectivity against an extensive range of dopamine, serotonin, adrenergic, histamine, and muscarinic receptors is described.
