126766-32-3 Usage
Description
GR 89696 FUMARATE is a selective κ-opioid receptor agonist, which possesses anti-nociceptive and neuroprotective properties. It is a pharmaceutical compound that has the potential to be used in various applications due to its ability to modulate the κ-opioid receptor.
Uses
Used in Pharmaceutical Industry:
GR 89696 FUMARATE is used as a pharmaceutical agent for its anti-nociceptive and neuroprotective properties. It is particularly useful in the development of treatments for pain management and neurodegenerative disorders.
Used in Pain Management:
GR 89696 FUMARATE is used as an analgesic agent for its ability to selectively activate the κ-opioid receptor, which is involved in pain modulation. This selective activation may provide effective pain relief with fewer side effects compared to traditional opioids.
Used in Neuroprotection:
GR 89696 FUMARATE is used as a neuroprotective agent due to its ability to protect neurons from damage and degeneration. This makes it a potential candidate for the treatment of neurodegenerative diseases such as Alzheimer's, Parkinson's, and multiple sclerosis.
Used in Drug Development:
GR 89696 FUMARATE is used as a research tool in the development of new drugs targeting the κ-opioid receptor. Its selective agonist properties make it valuable for studying the receptor's role in pain and neuroprotection, as well as for identifying potential therapeutic agents with improved efficacy and safety profiles.
Biological Activity
Highly potent and selective κ -opioid agonist (IC 50 = 0.04 nM) that may be selective for the putative κ 2 receptor. Anti-nociceptive and neuroprotective in vivo .
Check Digit Verification of cas no
The CAS Registry Mumber 126766-32-3 includes 9 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 6 digits, 1,2,6,7,6 and 6 respectively; the second part has 2 digits, 3 and 2 respectively.
Calculate Digit Verification of CAS Registry Number 126766-32:
(8*1)+(7*2)+(6*6)+(5*7)+(4*6)+(3*6)+(2*3)+(1*2)=143
143 % 10 = 3
So 126766-32-3 is a valid CAS Registry Number.
InChI:InChI=1/C19H25Cl2N3O3.C4H4O4/c1-27-19(26)23-8-9-24(15(13-23)12-22-6-2-3-7-22)18(25)11-14-4-5-16(20)17(21)10-14;5-3(6)1-2-4(7)8/h4-5,10,15H,2-3,6-9,11-13H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1+
