1310683-99-8Relevant articles and documents
Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors
Ettari, Roberta,Zappalà, Maria,Micale, Nicola,Grazioso, Giovanni,Giofrè, Salvatore,Schirmeister, Tanja,Grasso, Silvana
experimental part, p. 2058 - 2065 (2011/06/21)
The design, chemical synthesis, and enzymatic activity evaluation of a set of falcipain-2 inhibitors are reported. These compounds contain a proven peptidomimetic recognition motif based on a benzo[1,4]diazepin-2-one (1,4-BDZ) framework built on a dipepti