1407513-69-2Relevant articles and documents
Formylated polyamines as peptidomimetics
Javor, Sacha,Janowsky, Aaron,Johnson, Robert,Wolfrum, Katherine,Tadayoni-Rebek, Mitra,Rebek Jr., Julius
, p. 6580 - 6582 (2012)
A new construct for imitating a natural peptide ligand using a modified retro-inverso sequence is described. It is demonstrated through the synthesis of a peptidomimetic derived from the endogenous sequence of leucine enkephalin. The product was active at 400 nM and selective for μ-opioid receptors.