150651-04-0Relevant articles and documents
Synthesis and inhibiting activities of 1-peptidyl-2-haloacetyl hydrazines toward cathepsin B and calpains
Giordano, C,Calabretta, R,Gallina, C,Consalvi, V,Scandurra, R,et al.
, p. 297 - 311 (2007/10/02)
Twenty-four 1-peptidyl-2-haloacetyl hydrazines which can be considered azapeptide halomethanes were synthesized and tested as models of cathepsin B, calpain I and calpain II inhibitors.Reagents designed for cathepsin B inactivation include Z-Tyr, Z-Tyr(I)