1612872-85-1Relevant articles and documents
Method for preparing N-arylsulfonamide from indoline and arylsulfonamide
-
Paragraph 0036-0037, (2019/10/01)
The invention discloses a method for preparing N-arylsulfonamide from indoline and arylsulfonamide, belonging to the technical field of C-H bond activation and functionalization catalyzed by a transition metal. The method includes adding 1-acetyl indoline
Ruthenium-catalyzed C7 amidation of indoline C-H bonds with sulfonyl azides
Pan, Changduo,Abdukader, Ablimit,Han, Jie,Cheng, Yixiang,Zhu, Chengjian
, p. 3606 - 3609 (2014/04/03)
A ruthenium-catalyzed direct C7 amidation of indoline C-H bonds with sulfonyl azides was developed. This procedure allows the synthesis of a variety of 7-amino-substituted indolines, which are useful in pharmaceutical. The good functional tolerances, as well as the mild conditions, are prominent feature of this method.