20265-39-8

Basic information

• Product Name: 4-Amino-2-methoxypyridine
• Synonyms: 2-METHOXY-PYRIDIN-4-YLAMINE;4-AMINO-2-METHOXYPYRIDINE;2-METHOXY-4-AMINOPYRIDINE;2-Methoxypyridin-4-amine;2-Methoxy-pyridin-4-ylamine ,97%;2-Methoxy-4-pyridineamine;4-Amino-6-methoxypyridine;4-Amino-2-methoxypyridine ,97%
• CAS NO: 20265-39-8
• Molecular Formula: C₆H₈N₂O
• Molecular Weight: 124.14
• EINECS: -0
• Product Categories: Amines;blocks;Pyridines;Pyridine;Pyridine series;Boronic Acid
• Mol File: 20265-39-8.mol
• Article Data: 8

Chemical Properties

• Melting Point: 87-88°C
• Boiling Point: 271.7 °C at 760 mmHg
• Flash Point: 118.1 °C
• Appearance: /
• Density: 1.139 g/cm³
• Vapor Pressure: 0.00635mmHg at 25°C
• Refractive Index: 1.56
• Storage Temp.: Keep in dark place,Inert atmosphere,Room temperature
• PKA: 7.29±0.30(Predicted)
• CAS DataBase Reference: 4-Amino-2-methoxypyridine(CAS DataBase Reference)
• NIST Chemistry Reference: 4-Amino-2-methoxypyridine(20265-39-8)
• EPA Substance Registry System: 4-Amino-2-methoxypyridine(20265-39-8)

Safety Data

• Hazard Codes: Xi,Xn
• Statements: 22-36
• Safety Statements: 26
• WGK Germany: 3
• HazardClass: IRRITANT
• Hazardous Substances Data: 20265-39-8(Hazardous Substances Data)

Usage

Chemical Properties

Off-white solid

InChI:InChI=1/C6H8N2O/c1-9-6-4-5(7)2-3-8-6/h2-4H,1H3,(H2,7,8)

Upstream product

• 14395-39-2 2-methoxy-4-nitropyridine N-oxide 
• 14432-12-3 4-Amino-2-chloropyridine 
• 67-56-1 methanol 
• 1628-89-3 2-methoxypyridine 
• 20773-98-2 2-methoxypyridine N-oxide 
• 124-41-4 sodium methylate 
• 88511-26-6 2-iodo-pyridin-4-ylamine 

Downstream Products

• 72716-86-0 4-cyano-2-methoxypyridine 
• 100367-39-3 4-bromo-2-methoxypyridine 
• 408502-23-8 2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
• 849353-31-7 4-[(tert-butoxycarbonyl)amino]-2-methoxypyridine 
• 1018812-92-4 5-[[(2-methoxypyridin-4-yl)amino]methylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione 
• 1313547-55-5 N-(2-methoxypyridin-4-yl)-4-nitrobenzenesulfonamide 
• 88617-85-0 4-amino-N-(2-methoxy-pyridin-4-yl)-benzenesulfonamide 
• 1173699-31-4 AMG 337 
• 898561-71-2 C₁₁H₁₆N₂O₂ 
• 1620846-26-5 4-chloro-2-(4-fluoro-2-methylphenoxy)-N-(2-oxo-1,2-dihydropyridin-4-yl)benzamide 
• 1620846-13-0 2-(2,4-difluorophenoxy)-N-(2-oxo-1,2-dihydropyridin-4-yl)-4-(trifluoromethyl)benzamide 
• 1620847-67-7 2-fluoro-N-(2-methoxypyridin-4-yl)-4-(trifluoromethyl)benzamide 

Relevant articles and documents

NICOTINIC RECEPTOR COMPOUNDS

Provided herein are compounds and methods of preparation of compounds that are capable of functioning as agonists or antagonists of a nicotinic receptor. Also provided are pharmaceutical compositions comprising one or more of these compounds, which may further comprise one or more additional therapeutic agents. Further provided are methods of treatment of various conditions that may be responsive to such activity at the nicotinic receptors, such as nicotine dependence.

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