22280-95-1Relevant articles and documents
A concise synthesis of (±)-methoxyfumimycin ethyl ester
Zhou, Zhiwang,Hu, Yu,Wang, Bin,He, Xiaoru,Ren, Gang,Feng, Lihua
, p. 378 - 380 (2014)
The protecting-group-free synthesis of (±)-methoxyfumimycin ethyl ester, a potential bacterial peptide deformylase (PDF) inhibitor, is reported. The synthetic approach features a tandem Friedel-Crafts alkylation/lactonisation access as a key reaction to g
Design, synthesis, characterization, and anticancer activity of a novel series of O-substituted chalcone derivatives
Ngameni, Bathélémy,Cedric, Kamdoum,Mbaveng, Armelle T.,Erdo?an, Musa,Simo, Ingrid,Kuete, Victor,Da?tan, Arif
, (2021)
A new series of O-substituted chalcone derivatives bearing an/a allyl-, prenyl- or propargyl-substituent at different positions of rings A and B and their derivatives as drug leads, was designed, synthesized, and characterized. The chalcone derivatives we
Introducing the Tishchenko reaction into sustainable polymer chemistry
Ren, Tianhua,Chen, Qin,Zhao, Changbo,Zheng, Qiang,Xie, Haibo,North, Michael
, p. 1542 - 1547 (2020)
Taking advantage of the structural characteristics of lignin-derived phenolic compounds, a combination of the Williamson and Tishchenko reactions produced a series of new α,ω-diene functionalized carboxylic ester monomers from both petrochemical and renewable resources, which were applicable in subsequent thiol-ene click and acyclic diene metathesis (ADMET) polymerizations, providing a series of poly(thioether esters) and unsaturated aromatic-aliphatic polyesters with high molecular weights.
Synthesis of the intermediate for fumimycin: A natural peptide deformylase inhibitor
Zhou, Zhi-Wang,Li, Wei-Chao,Hu, Yu,Wang, Bin,Ren, Gang,Feng, Li-Hua
, p. 3049 - 3054 (2013)
Synthetic efforts toward the potential bacterial peptide deformylase inhibitor fumimycin are reported. The synthetic approach features a tandem Friedel-Crafts alkylation/lactonization access as key reaction to the α, α-disubstituted amino acid unit, and r
Iodine-DMSO catalyzed chemoselective oxidative aromatization and deallylation, nondeallylation of aryl allyl ether of tetrahydro-β-carboline
Gaikwad, Sunil V.,Gaikwad, Milind V.,Lokhande, Pradeep D.
supporting information, p. 1408 - 1414 (2021/04/26)
We have developed a simple method for the chemoselective aromatization of tetrahydro-β-carboline with selective nondeallylation O-allyl groups in the presence of iodine (100 mol %) in dimethyl sulfoxide/H2O2. A convergent approach toward the oxidative aromatization with selective deallylation (deprotection) of O-allyl-tetrahydro-β-carboline using iodine in dimethyl sulfoxide/HCl has been described. The present protocol contains cheap catalyst, easy work up, normal reaction conditions, and high selectivity.