27065-51-6Relevant articles and documents
IMINO SULFANONE INHIBITORS OF ENPP1
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Paragraph 0205, (2021/11/13)
The present disclosure relates generally to inhibitors of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1), compositions thereof, and methods of using said compounds and compositions thereof. More specifically, the present disclosure relates to sulfoximine- based inhibitors of ENPP1 of Formula (I) and methods of their use for treating disease mediated by ENPP1.
Synthesis of substituted bis(heteroaryl)maleimides
Dubernet, Mathieu,Caubert, Virginie,Guillard, Jér?me,Viaud-Massuard, Marie-Claude
, p. 4585 - 4593 (2007/10/03)
Substituted bis(fur-2-yl), bis(fur-3-yl) and bis(thien-2-yl) maleimides with potential antidiabetic properties are described. Their synthesis involves, as a key step, a Suzuki cross-coupling between various boron derivatives and the diiodomaleimides. Therefore, a wide range of substituted symmetric and non-symmetric maleimide derivatives can be prepared.
Synthetic routes to cristatic acid and derivatives
Chiarello,Joullie
, p. 41 - 48 (2007/10/02)
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