60295-18-3Relevant articles and documents
Oxaziridine-mediated amination of primary amines: Scope and application to a one-pot pyrazole synthesis
Armstrong, Alan,Jones, Lyn H.,Knight, Jamie D.,Kelsey, Richard D.
, p. 713 - 716 (2007/10/03)
(Chemical Equation Presented) Electrophilic amination of primary aliphatic and aromatic amines is reported using a diethylketomalonate-derived oxaziridine to afford the corresponding N-Boc hydrazines in good to excellent yields. The method allows a one-pot synthesis of pyrazoles from primary amines.