857775-99-6Relevant articles and documents
Mild and efficient synthesis of indoles and isoquinolones via a nickel-catalyzed Larock-type heteroannulation reaction
Weng, Wei-Zhi,Xie, Jian,Zhang, Bo
supporting information, p. 3983 - 3988 (2018/06/08)
A simple and efficient approach for the preparation of substituted indoles and isoquinolones via a nickel-catalyzed Larock-type heteroannulation reaction is reported. This transformation employed air-stable and inexpensive Ni(dppp)Cl2 as a precatalyst and Et3N as a mild base. Moreover, the reaction occurs efficiently under mild conditions, and a wide range of substituted indoles and isoquinolones bearing various functional groups are obtained in moderate to excellent yields.
Synthesis of indoles and polycyclic amides via ruthenium(ii)-catalyzed C-H activation and annulation
Lin, Hui,Li, Shuai-Shuai,Dong, Lin
supporting information, p. 11228 - 11234 (2015/11/27)
Ruthenium(ii)-catalyzed oxidative coupling of NH protic amides with alkynes has been developed for the synthesis of a diversity of complex structures, such as N-acyl indole and tricyclic amide derivatives.
Synthesis of indoles via palladium-catalyzed C-H activation of N-aryl amides followed by coupling with alkynes
Zhou, Feng,Han, Xiuling,Lu, Xiyan
, p. 4681 - 4685 (2011/09/30)
A convenient and efficient method for the construction of indole skeleton was developed via Pd-catalyzed C-H activation of N-aryl amides and subsequent coupling with alkynes. Both stoichiometric and catalytic versions have been successfully achieved.
