863640-20-4Relevant articles and documents
Novel 3-amino-2-hydroxy acids containing protease inhibitors. Part 1: Synthesis and kinetic characterization as aminopeptidase P inhibitors
Stoeckel-Maschek, Angela,Stiebitz, Beate,Koelsch, Regine,Neubert, Klaus
, p. 4806 - 4820 (2007/10/03)
Novel, potent inhibitors of aminopeptidase P, containing a 3-amino-2-hydroxy acid and a proline or a proline analogues, have been prepared. One part of the bestatin-derived inhibitors was found to inhibit APP from Escherichia coli and from rat intestine a