Bioisosteric heterocyclic versions of 7-{[2-(4-phenyl-piperazin-1-yl)ethyl] propylamino}-5,6,7,8-tetrahydronaphthalen-2-ol: Identification of highly potent and selective agonists for dopamine D3 receptor with potent in vivo activity
In the current report, we extend the SAR study on our hybrid structure 7-{[2-(4-phenyl-piperazin-1-yl)ethyl]propylamino}-5,6,7,8-tetrahydronaphthalen- 2-ol further to include heterocyclic bioisosteric analogues. Binding assays were carried out with HEK-29
Biswas, Swati,Hazeldine, Stuart,Ghosh, Balaram,Parrington, Ingrid,Kuzhikandathil, Eldo,Reith, Maarten E. A.,Dutta, Aloke K.
experimental part
p. 3005 - 3019
(2009/04/06)
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