cas 112904-74-2, 8-hydroxy-3,4-dihydro-3-(dipropylamino)-2H-1-benzopyran

Articles about 112904-74-2Total 2 be found

Methoxy and hydroxy derivatives of 3,4-dihydro-3-(di-n-propylamino)-2H-1-benzopyrans: New synthesis and dopaminergic activity
The synthesis of methoxy and hydroxy derivatives of 3,4-dihydro-3-(di-n-propylamino)-2H-1-benzopyran from readily available or commercial o-hydroxybenzaldehydes is described in six steps. The enantiomers of 8-hydroxy-3,4-dihydro-3-(di-n-propyl-amino)-2H-1-benzopyran 1b have been resolved. It is shown that the compound (-)-1b is a mroe selective D-2 agonist, compared to apomorphine.
Al Neirabeyeh,Reynaud,Podona,Ou,Perdicakis,Coudert,Guillaumet,Pichat,Gharib,Sarda
p. 497 - 504
(2007/10/02)

Synthesis and dopaminergic activity of a new oxygen isostere of the 2-aminotetralins: N,N-dipropyl-8-hydroxy-3-chromanamine
The synthesis of N,N-dipropyl-8-hydroxy-3-chromanamine from 8-methoxy-4-chromanone oxime in seven steps is described.This compound is an oxygen isostere of the dopamine (DA) receptor agonist N,N-dipropyl-5-hydroxy-2-aminotetralin.In in vitro and in vivo t
Horn, Alan S.,Kaptein, Bernard,Vermue, Niek A.,Vries, Jan B. De,Mulder, Theo B. A.
p. 325 - 328
(2007/10/02)