- Structure-activity evaluation of n-benzyl-5-substituted indole-3-imine derivatives and their amine congeners as bovine testicular hyaluronidase (BTH) inhibitor
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With the aim to overcome the lack of potent and selective Hyaluronidases (Hyals) inhibitors, we have tested new 1, 3 and 5 substituted indole derivatives for the inhibition of bovine testicular hyaluronidases (BTH) in a stains-all assay at pH 7 and in a M
- Oelgen,Kaessler,Kilic Kurt,Jose
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scheme or table
p. 685 - 690
(2012/04/05)
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- Synthesis and pp60c-Src tyrosine kinase inhibitory activities of novel indole-3-imine and amine derivatives substituted at N1 and C5
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A series of novel 1,3,5-trisubstituted indole derivatives, namely, N-benzyl 5-phenyl indole-3-imine, N-benzyl-5-(p-fluorophenyl)indole-3-imine and their corresponding amine congeners, were designed and synthesized as pp60 c-Src tyrosine kinase
- Kilic, Zuhal,Isgoer, Yasemin G.,Oelgen, Suereyya
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experimental part
p. 333 - 343
(2009/10/24)
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