BENZO[d]OXAZOLES AND BENZO[d]THIAZOLES AS KINASE INHIBITORS
Novel benzo[d]oxazole and/or benzo[d]thiazole compounds, pharmaceutical compositions containing the benzo[d]oxazole and/or benzo[d]thiazole compounds, and methods of their pharmaceutical use are disclosed. In certain embodiments, the benzo[d]oxazole and/o
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(2010/04/06)
Benzothiazoles as Rho-associated kinase (ROCK-II) inhibitors
A series of benzothiazole derivatives as ROCK inhibitors have been discovered. Compounds with good biochemical and cellular potency, and sufficient kinase selectivity have been identified.