Photoredox-catalyzed deuteration and tritiation of pharmaceutical compounds
Deuterium- and tritium-labeled pharmaceutical compounds are pivotal diagnostic tools in drug discovery research, providing vital information about the biological fate of drugs and drug metabolites. Herein we demonstrate that a photoredox-mediated hydrogen
Loh, Yong Yao,Nagao, Kazunori,Hoover, Andrew J.,Hesk, David,Rivera, Nelo R.,Colletti, Steven L.,Davies, Ian W.,MacMillan, David W. C.
p. 1182 - 1187
(2017/12/08)
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