1266317-80-9Relevant articles and documents
Enantioselective synthesis of 3-substituted tryptamines as core components of central nervous system drugs and indole natural products
Hanessian, Stephen,Stoffman, Elia J.L.
, p. 13 - 20 (2013/03/13)
Application of the MacMillan iminium ion Michael and Friedel-Crafts type reactions to γ-amino α,β-unsaturated butanals led to the corresponding β-substituted butanals in good yields and high enantioselectivities. The products could be useful intermediates
Applications of organocatalytic asymmetric synthesis to drug prototypes-dual action and selective inhibitors of n -nitric oxide synthase with activity against the 5-HT1D/1B subreceptors
Hanessian, Stephen,Stoffman, Eli,Mi, Xueling,Renton, Paul
scheme or table, p. 840 - 843 (2011/04/27)
The scope of MacMillan's organocatalytic asymmetric conjugate addition reaction of indoles and electron-rich aromatics to α,β-unsaturated aldehydes has been extended to the use of 3-amino crotonaldehydes as substrates. The aromatics used include indoles a
