1313388-99-6Relevant academic research and scientific papers
New 2-heterocyclyl-imidazo[2,1- i ]purin-5-one derivatives as potent and selective human A3 adenosine receptor antagonists
Baraldi, Pier Giovanni,Preti, Delia,Zaid, Abdel Naser,Saponaro, Giulia,Tabrizi, Mojgan Aghazadeh,Baraldi, Stefania,Romagnoli, Romeo,Moorman, Allan R.,Varani, Katia,Cosconati, Sandro,Di Maro, Salvatore,Marinelli, Luciana,Novellino, Ettore,Borea, Pier Andrea
experimental part, p. 5205 - 5220 (2011/10/08)
A series of 4-allyl/benzyl-7,8-dihydro-8-methyl/ethyl-2-[(substituted) isoxazol/pyrazol-3/5-yl]-1H-imidazo[2,1-i]purin-5(4H)-ones has been synthesized and evaluated in radioligand binding assays to determine their affinities at the human A1, A
