Novel vitamin D receptor ligands bearing a spherical hydrophobic core structure-Comparison of bicyclic hydrocarbon derivatives with boron cluster derivatives
Vitamin D receptor (VDR) is a nuclear receptor for 1a,25-dihydroxyvitamin D3 (1a,25(OH)2D3), and is an attractive target for multiple clinical applications. We recently developed novel non-secosteroidal VDR ligands bearing a hydrophobic p-carborane cage,
Wongmayura, Angsuma,Fujii, Shinya,Ito, Shigeru,Kano, Atsushi,Taoda, Yoshiyuki,Kawachi, Emiko,Kagechika, Hiroyuki,Tanatani, Aya
p. 1756 - 1760
(2012/04/04)
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