2-(4-Methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure-activity relationships in the B and C-regions
On the basis of the previous lead N-4-t-butylbenzyl 2-(3-fluoro-4- methylsulfonylaminophenyl) propanamide (3) as a potent TRPV1 antagonist, structure-activity relationships for the B (propanamide part) and C-region (4-t-butylbenzyl part) have been investi
Sun, Wei,Liu, Keliang,Ryu, Hyungchul,Kang, Dong Wook,Kim, Yong Soo,Kim, Myeong Seop,Cho, Yongsung,Bhondwe, Rahul S.,Thorat, Shivaji A.,Kim, Ho Shin,Pearce, Larry V.,Pavlyukovets, Vladimir A.,Tran, Richard,Morgan, Matthew A.,Lazar, Jozsef,Ryder, Christopher B.,Toth, Attila,Blumberg, Peter M.,Lee, Jeewoo
experimental part
p. 1310 - 1318
(2012/04/04)
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