136689-94-6Relevant articles and documents
Zinc hydroxyapatite - Catalyzed efficient synthesis of 5-substituted 1H-tetrazoles
Lakshmi Kantam,Balasubrahmanyam,Shiva Kumar
, p. 1809 - 1814 (2006)
Zinc hydroxyapatite (ZnHAP) is an effective heterogeneous catalyst for the (2 + 3)-cycloaddition of sodium azide with nitriles to afford 5-substituted 1H-tetrazoles in good yields. The catalyst is recovered and reused for several cycles with consistent ac
Microwave assisted synthesis of novel tetrazole/sulfonamide derivatives based on octahydroacridine, xanthene and chromene skeletons as inhibitors of the carbonic anhydrases isoforms I, II, IV and VII
Esirden, ?brahim,Tan?, Muhammet,Supuran, Claudiu T.,Kaya, Muharrem
, p. 86 - 89 (2017)
The synthesis of novel tetrazole/sulfonamide derivatives based on octahydroacridine, xanthene and chromene scaffold by using microwave (MW) assisted techniques is reported in this study. These synthesized hybrid compounds were assayed for the inhibition o
Facile, highly efficient and novel method for synthesis of 5-substituted 1H-tetrazoles catalysed by copper(I) chloride
Esirden, Ibrahim,Ba?ar, Erhan,Kaya, Muharrem
, p. 1231 - 1236 (2015)
The present study on tetrazole compounds, which have a wide area of application, proposes a new, simple and highly effective method. A series of 5-substituted 1H-tetrazoles were synthesised in DMF via the [3 + 2] cycloaddition reaction, in which different
One-pot synthesis of 5-substituted lH-tetrazoles from aryl bromides with potassium hexakis(cyano-κC)ferrate(4 -)(K4[Fe(CN)6]) as cyanide source
Zhu, Yizhong,Ren, Yiming,Cai, Chun
, p. 171 - 175 (2009)
A one-pot procedure for the synthesis of 5-substituted 1H-tetrazoles through the three-component reaction between an aryl bromide, potassium hexakis(cyano-κC)ferrate(4 - ) (K4[Fe(CN)6]) and NaN3 catalyzed by [Pd(OAc)2
Design, synthesis and evaluation of 1,3,6-trisubstituted-4-oxo-1,4-dihydroquinoline-2-carboxylic acid derivatives as ETA receptor selective antagonists using FRET assay
Khadtare, Nikhil,Stephani, Ralph,Korlipara, Vijaya
, p. 2281 - 2285 (2017/05/10)
The endothelin axis and in particular the two receptor subtypes, ETA and ETB, are under investigation for the treatment of various diseases such as pulmonary arterial hypertension, fibrosis, renal failure and cancer. Previous work in
Synthesis of 5-substituted-1H-tetrazole derivatives using monodisperse carbon black decorated Pt nanoparticles as heterogeneous nanocatalysts
Baskaya, Gaye,Esirden, Ibrahim,Erken, Esma,Sen, Fatih,Kaya, Muharrem
, p. 1992 - 1999 (2017/01/28)
A facile and highly efficient protocol for synthesis of new 5-substituted 1H-tetrazoles derivatives has been developed by the assistance of vulcan carbon decorated based on monodisperse platinum nanoparticles (Pt NPs@VC) as superior and recyclable heterog
Identification of a New Class of Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors Followed by a Structure-Activity Relationship Study
Hansen, Stinne W.,Erichsen, Mette N.,Fu, Bingru,Bj?rn-Yoshimoto, Walden E.,Abrahamsen, Bjarke,Hansen, Jacob C.,Jensen, Anders A.,Bunch, Lennart
, p. 8757 - 8770 (2016/10/22)
Screening of a small compound library at the three excitatory amino acid transporter subtypes 1-3 (EAAT1-3) resulted in the identification of compound (Z)-4-chloro-3-(5-((3-(2-ethoxy-2-oxoethyl)-2,4-dioxothiazolidin-5-ylidene)methyl)furan-2-yl)benzoic aci
RETRACTED ARTICLE: A rapid and novel method for the synthesis of 5-substituted 1H-tetrazole catalyzed by exceptional reusable monodisperse Pt NPs@AC under the microwave irradiation
Erken, Esma,Esirden, Ibrahim,Kaya, Muharrem,Sen, Fatih
, p. 68558 - 68564 (2015/09/01)
A series of 5-substituted 1H-tetrazoles were synthesized in DMF by the [3 + 2] cycloaddition reaction under the effect of microwave irradiation (10-30 min, fixed mode, 90 °C, 140 W) in the presence of highly efficient superior catalyst. For this reaction,
RETRACTED ARTICLE: Monodisperse Pt NPs@rGO as highly efficient and reusable heterogeneous catalysts for the synthesis of 5-substituted 1H-tetrazole derivatives
Esirden, Ibrahim,Erken, Esma,Kaya, Muharrem,Sen, Fatih
, p. 4452 - 4457 (2015/09/01)
Monodisperse platinum nanoparticles supported on reduced graphene oxide (Pt NPs@rGO) are stable, isolable, bottleable, long-lived, highly efficient and exceptionally reusable heterogeneous catalysts for the synthesis of 5-substituted 1H-tetrazoles from so
Thiosemicarbazones of formyl benzoic acids as novel potent inhibitors of estrone sulfatase
Jütten, Peter,Schumann, Winfried,H?rtl, Albert,Dahse, Hans-Martin,Gr?fe, Udo
, p. 3661 - 3666 (2008/02/11)
Thiosemicarbazones of the microbial metabolite madurahydroxylactone, a polysubstituted benzo[a]-naphthacenequinone, have been previously reported by us as potent nonsteroidal inhibitors of the enzyme estrone sulfatase (cyclohexylthiosemicarbazone 1, ICsu
