137858-18-5Relevant articles and documents
Amino substituted pyrimido[1,6-2]benzimidazoles
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, (2008/06/13)
The present invention relates to novel substituted pyrimidobenzimidazole derivatives of the formula STR1 wherein the substituents are as described in the specification, and pharmaceutically acceptable salts thereof. The products have an inhibitory action
Pyrimido[1,6-a]benzimidazoles: A new class of DNA gyrase inhibitors
Hubschwerlen,Pflieger,Specklin,Gubernator,Gmunder,Angehrn,Kompis
, p. 1385 - 1392 (2007/10/02)
Substituted 4-quinolone- (1, A = CH) and 1,8-naphthyrid-4-one- (1, A = N) 3-carboxylic acids are currently the only classes of clinically useful antibacterial agents exerting their activity by inhibiting the subunit A of DNA gyrase. Pyrimido[1,6-a]benzimi