- 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF
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The present invention provides compounds, compositions thereof, and methods of using the same.
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Paragraph 00329
(2017/09/27)
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- PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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This document discloses molecules having the following formula (“Formula One”): and processes related thereto.
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Paragraph 0622; 0623
(2016/05/02)
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- PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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This document discloses molecules having the following formula (“Formula One”): and processes related thereto.
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Paragraph 0622-0623
(2013/11/06)
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- BICYCLIC -AMINO ACID DERIVATIVE
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It is intended to provide a bicyclic γ-amino acid derivative having excellent activity as an α2δ ligand. The present invention provides a compound represented by the general formula (I): wherein R1, R2, R2', R4, R5, R6, R7, R8, and R8' are a hydrogen atom or the like; and R3 is a hydrogen atom, a halogen atom, a C1-C6 alkyl group, or the like.
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Page/Page column 52; 53
(2010/06/17)
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- SUBSTITUTED BENZOFUSED DERIVATIVES AND THEIR USE AS VANILLOID RECEPTOR LIGANDS
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The present invention relates to substituted benzofused derivatives, which can be used as vanilloid receptor ligands, method of treating diseases, conditions and/or disorders modulated by vanilloid receptors with them, and processes for preparing them.
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Page/Page column 34
(2010/11/27)
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- Rearrangement of isoxazoline-5-spiro derivatives. Part 7. Thermal rearrangement of 4,5-dihydro and tetrahydroisoxazole-5-spirocyclobutanes to azepin-4-one derivatives
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Some representative 4,5-dihydro and tetrahydroisoxazole-5-spirocyclobutanes have been synthesized by 1,3-dipolar cycloaddition of alkylidenecyclobutanes to nitrile oxides and nitrones, respectively. When subjected to flash vacuum thermolysis conditions, the spiranic cycloadducts rearranged to afford mainly the desired azepin-4-one derivatives. In addition, the isoxazoline cycloadducts gave unexpected by-products, which were identified as 1-alkenyl-2-pyrrolidinones. Analogies and differences with respect to the lower homologue cyclopropanes are evidenced in both cycloaddition and rearrangement reactions.
- Goti,Brandi,De Sarlo,Guarna
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p. 5283 - 5300
(2007/10/02)
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