152241-38-8Relevant articles and documents
GAMMA-AMINOAMIDE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY
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Page/Page column 71, (2010/02/07)
The present invention is directed to compounds of the formula (I), wherein R1, R2, R3, R4, R5, R6, R7, R8, R11, R12, W, X, and n are defined herein, which are useful as modulators of chemokine receptor activity. In particular, these compounds are useful as modulators of the chemokine receptor CCR-2.
4-[4'-PIPERODINYL OR 3'-PIRROLIDINYL] SUBSTITUTED IMIDAZOLES AS H3 RECEPTOR ANTAGONISTS AND THERAPEUTIC USES THEREOF
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, (2008/06/13)
Diazolyl compounds having activity as histamine H3-receptor antagonists, pharmaceutical compositions and methods of using such compounds for treating cognitive disorder or attention or arousal deficit.
HISTAMINE H3-RECEPTOR ANTAGONISTS AND THERAPEUTIC USES THEREOF
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, (2008/06/13)
The present invention is directed to compounds of the class of piperidyl-imidazole derivative histamine H 3-receptor antagonists. Such compounds have affinity for histamine H 3-receptor, and preferably penetrate the blood-brain barrier. The compounds can
Process for the preparation of intermediates useful for the synthesis of histamine receptor antagonists
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, (2008/06/13)
The present invention relates to a novel process for the preparation of highly potent histamine receptor antagonists, in particular histamine H 3 receptor antagonists. Also disclosed is a novel process for the preparation of intermediates useful in the preparation of histamine receptor antagonists, in particular H 3 -receptor antagonists.