Bronsted acid-promoted sequential hydroarylation-hydroamidation of arene-tethered 1-(2-alkynylphenyl)ureas: Direct access to 4,4-spiro-3,4-dihydro- 2-(1H)-quinazolinones
A Bronsted acid-promoted approach to 4,4-sipro-3,4-dihydro-2-(1H)- quinazolinones from arene-tethered 1-(2-alkynylphenyl)ureas has been developed. The reaction is initiated by intramolecular hydroarylation followed by hydroamidation, assisted by intramole
Cinnolines and Pyrazolopyridazines. - Novel Synthetic and Mechanistic Aspects of the Richter Reaction
The thermal cyclization of 2-alkynylbenzenediazonium salts 2 known as the Richter reaction and leading, as described in the literature, only to 4-hydroxycinnolines 6 has been studied.A new probable route to these compounds involving intermediate formation
Vasilevsky, Sergei F.,Tretyakov, Eugene V.
p. 775 - 780
(2007/10/02)
More Articles about upstream products of 157869-09-5