Direct amination of pyrimidin-2-yl tosylates with aqueous ammonia under metal-free and mild conditions
Abstract A metal-free synthesis of pyrimidine functionalized primary amines via direct amination of pyrimidin-2-yl tosylate with aqueous ammonia has been developed under mild conditions. The desired products pyrimidin-2-amines can be generated in excellen
A process for the preparation of a compound of Formula (1) and intermediates useful therein are provided. The process comprises reacting a compound of formula R1-CO-CH2-E with a compound of formula R2-CHX1X
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Page 8
(2008/06/13)
Process for preparing 2-amino-4-(4-fluorphenyl)-6-alkylpyrimidine-5-carboxylate
A process for the preparation of a compound of the formula: wherein the variables are herein below defined.
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(2008/06/13)
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