Preparation of carbon-14 labeled 3,4-dihydro-5-methyl-1(2H)-isoquinolinone
Carbon-14 labeled 3,5-dihydro-5-methyl-1(2H)-isoquinolinone, a potent inhibitor of poly(ADP-ribose) polymerase (ADPRP) was prepared from 1-bromo-2-methylbenzene in 7.8 % overall yield. The C-14 label was introduced from Ba(l)4CO3 via
Ekhato,Huang
p. 627 - 634
(2007/10/02)
More Articles about upstream products of 24080-02-2