Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1'-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1'-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines
Few muscarinic antagonists differentiate between the M4 and M2 muscarinic receptors. In a structure-activity study, aimed at discovering leads for the development of a M4 muscarinic receptor-selective antagonist, we have s
Manfredini, Stefano,Lampronti, Ilaria,Vertuani, Silvia,Solaroli, Nicola,Recanatini, Maurizio,Bryan, David,Mckinney, Michael
p. 1559 - 1566
(2007/10/03)
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