- AMIDINOANILINE DERIVATIVE
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Provided are a novel amidine derivative having an activated blood coagulation factor X inhibitory activity, a production method thereof, a production intermediate therefor, and a pharmaceutical composition containing the amidine derivative. An amidinoanil
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Paragraph 0176-0179; 0212-0214
(2013/03/26)
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- Inhibitors of factor Xa
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Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.
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Page column 199
(2010/02/05)
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- Cyclic amino acid derivatives
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Novel compounds of the formula I 1in which R1, R2, R2′, R2″, R3, R4, R5, R5′, R5″, R5′″, R5″″, X, Y, U, V and W are as defined in Patent claim 1, are inhibitors of coagulation factors Xa and VIIa and can be employed fr the treatment of thromboses, myocardilal infarction, arteriosclerosis, inflammation, apoplexia, angina pectoris, restenosis after angioplasty, claudicatio intermittens, tumours, tumour diseases and/or tumour metastases.
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